• Product NamePerphenazine
• Brief DescriptionInhibitors
• Purification99.30%
• Biological ActivityPerphenazine is a typical antipsychotic drug, inhibits 5-HT2A receptor (5-HT2A), Alpha-1A adrenergic receptor (α1A), Dopamine receptor D2/D3, D2L receptor, and Histamine H1 receptor (H1) with Ki of 5.6, 10, 0.765/0.13, 3.4, and 8 nM.
• Target NameCaMK inhibitor; Dopamine Receptor antagonist
• CAS No. 58-39-9
• Calculated MW 403.97
• Formulation C21H26ClN3OS
• Storage 3 years -20˚C powder;2 years -80˚C in solvent;

• Research Area:Nervous system
  SMILES:OCCN1CCN(CCCN2C3=CC=CC=C3SC3=C2C=C(Cl)C=C3)CC1
  Pathways:GPCR/G Protein; Neuroscience
  Receptor:CAM; Dopamine
  Boling pt:580.4C?
  Melting pt:35339C
  Solubility:Soluble in DMSO
  Appearance:White Powder
  Remark:For obtaining a higher solubility , please warm the tube at 37 ˚C and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ˚C for several month.

1. Hoyberg OJ, et al. Acta Psychiatr Scand. 1993 Dec;88(6):395-402.

• Flow Cytometry (FCM) General Protocol
• Immunofluorescence(IC)
• Immunohistochemistry(Polymer)
• Western Blotting