• Product NameAzasetron hydrochloride
• Brief DescriptionInhibitors
• Purification99.50%
• Biological ActivityAzasetron Hydrochloride is a 5-HT3 receptor antagonist which is used as an anti-emetic.Azasetron inhibited the specific binding of [3H]quipazine to 5-HT3 receptors at the synaptic membranes of the rat cerebral cortex.
• Target Name5-HT Receptor antagonist
• CAS No. 123040-16-4
• Calculated MW 386.27
• Formulation C17H20ClN3O3HCl
• Storage 3 years -20˚C powder;2 years -80˚C in solvent;

• Research Area:Nervous system
  SMILES:Cl.CN1C(=O)COC2=C1C=C(Cl)C=C2C(=O)NC1CN2CCC1CC2
  Pathways:GPCR/G Protein; Neuroscience
  Receptor:5-HT3
  Boling pt:558C?
  Melting pt:
  Solubility:Water: 3 mg/mL (7.76 mM)
  Appearance:White Powder
  Remark:For obtaining a higher solubility , please warm the tube at 37 ˚C and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ˚C for several month.

1. Katayama K, et al. Jpn J Pharmacol. 1997 Apr;73(4):357-60.

• Flow Cytometry (FCM) General Protocol
• Immunofluorescence(IC)
• Immunohistochemistry(Polymer)
• Western Blotting