• Product NameGSK503
• Brief DescriptionInhibitors
• Purification98.00%
• Biological ActivityGSK-503 is a potent EZH2 inhibitor with potential antiY activity.
• Target NameHistone Methyltransferase inhibitor
• CAS No. 1346572-63-1
• Calculated MW 526.67
• Formulation C31H38N6O2
• Storage 3 years -20˚C powder;2 years -80˚C in solvent;

• Research Area:Other
  SMILES:CC(C)N1C=C(C)C2=C(C=C(C=C12)C1=CN=C(C=C1)N1CCN(C)CC1)C(=O)NCC1=C(C)C=C(C)NC1=O
  Pathways:Chromatin/Epigenetic
  Receptor:EZH2
  Boling pt:
  Melting pt:
  Solubility:Ethanol: 26 mg/mL warmed (49.36 mM); DMSO: 100 mg/mL (189.87 mM)
  Appearance:White Powder
  Remark:For obtaining a higher solubility , please warm the tube at 37 ˚C and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ˚C for several month.

1. Zingg D, et al. Nat Commun. 2015 Jan 22;6:6051.

• Flow Cytometry (FCM) General Protocol
• Immunofluorescence(IC)
• Immunohistochemistry(Polymer)
• Western Blotting