• Product NameOtenabant (CP-945598) hydrochloride
• Brief DescriptionInhibitors
• Purification99.52%
• Biological ActivityOtenabant hydrochloride (CP-945598) is a recently discovered selective, high affinity, competitive CB1 receptor antagonist with Ki of 0.7 nM.
• Target NameCannabinoid Receptor antagonist
• CAS No. 686347-12-6
• Calculated MW 546.88
• Formulation C25H26Cl3N7O
• Storage 3 years -20˚C powder;2 years -80˚C in solvent;

• Research Area:Other
  SMILES:CCNC1(CCN(CC1)C1=NC=NC2=C1NC(N2C1=CC=C(Cl)C=C1)C1=CC=CC=C1Cl)C(N)=O
  Pathways:GPCR/G Protein
  Receptor:hCB1; hCB2; rCB1
  Boling pt:
  Melting pt:
  Solubility:DMSO: 1 mg/mL warmed (1.82 mM)
  Appearance:White Crystalline Powder
  Remark:For obtaining a higher solubility , please warm the tube at 37 ˚C and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ˚C for several month.

1. John R. Hadcock, et al. Biochemical and Biophysical Research Communications,2010; 394;366-371.

• Flow Cytometry (FCM) General Protocol
• Immunofluorescence(IC)
• Immunohistochemistry(Polymer)
• Western Blotting