• Product NameWH-4-023
• Brief DescriptionInhibitors
• Purification99.75%
• Biological ActivityWH-4-023 is a potent and orally active Lck/Src inhibitor with IC50 of 2 nM and 6 nM in cell-free assays, respectively.
• Target NameSrc inhibitor
• CAS No. 837422-57-8
• Calculated MW 568.67
• Formulation C32H36N6O4
• Storage 3 years -20˚C powder;2 years -80˚C in solvent;

• Research Area:Other
  SMILES:COC1=CC(OC)=C(C=C1)N(C(=O)OC1=C(C)C=CC=C1C)C1=NC(NC2=CC=C(C=C2)N2CCN(C)CC2)=NC=C1
  Pathways:Angiogenesis
  Receptor:Lck; Src
  Boling pt:
  Melting pt:
  Solubility:Ethanol: 6 mg/mL warmed (10.55 mM); DMSO: 12 mg/mL warmed (21.1 mM)
  Appearance:White Powder
  Remark:For obtaining a higher solubility , please warm the tube at 37 ˚C and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ˚C for several month.

1. Martin MW, et al. J Med Chem. 2006 Aug 10;49(16): 4981-91.

• Flow Cytometry (FCM) General Protocol
• Immunofluorescence(IC)
• Immunohistochemistry(Polymer)
• Western Blotting