- Product NamePFI-2
- Brief DescriptionInhibitors
- Purification99.91%
- Biological ActivityPFI-2 is a potent, selective, and cell-active lysine methyltransferase SETD7 inhibitor with Ki (app) and IC50 of 0.33 nM and 2 nM, 1000-fold selectivity over other methyltransferases and other non-epigenetic targets.
- Target NameHistone Methyltransferase inhibitor
- CAS No. 1627676-59-8
- Calculated MW 499.52
- Formulation C23H25F4N3O3S
- Storage 3 years -20˚C powder;2 years -80˚C in solvent;