• Product NameCNV-1014802
• Brief DescriptionInhibitors
• Purification98.00%
• Biological ActivityCNV1014802(GSK-1014802) is a novel small molecule state-dependent sodium channel blocker; Nav1.7 sodium channel inhibitor.
• Target NameSodium Channel inhibitor
• CAS No. 934240-30-9
• Calculated MW 314.35
• Formulation C18H19FN2O2
• Storage 3 years -20˚C powder;2 years -80˚C in solvent;

• Research Area:Cancer
  SMILES:C1C[C@H](N[C@H]1C2=CC=C(C=C2)OCC3=CC=CC=C3F)C(=O)N
  Pathways:Membrane transporter/Ion channel
  Receptor:Sodium Channel
  Boling pt:
  Melting pt:
  Solubility:DMSO: 10 mM
  Appearance:White Powder
  Remark:For obtaining a higher solubility , please warm the tube at 37 ˚C and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ˚C for several month.

1. Large CH, et al. J Pharmacol Exp Ther. 2011 Jul;338(1):100-13.

• Flow Cytometry (FCM) General Protocol
• Immunofluorescence(IC)
• Immunohistochemistry(Polymer)
• Western Blotting