• Product NameGSK2801
• Brief DescriptionInhibitors
• Purification98.00%
• Biological ActivityGSK2801 is a potent, selective and cell active acetyl-lysine competitive inhibitor of BAZ2A(Kd=136 nM) and BAZ2B(Kd=257 nM) bromodomains.
• Target NameEpigenetic Reader Domain inhibitor
• CAS No. 1619994-68-1
• Calculated MW 371.45
• Formulation C20H21NO4S
• Storage 3 years -20˚C powder;2 years -80˚C in solvent;

• Research Area:Cancer
  SMILES:CCCOC1=CC2=C(C=C(N2C=C1)C(C)=O)C1=CC=CC=C1S(C)(=O)=O
  Pathways:Chromatin/Epigenetic
  Receptor:BAZ2A; BAZ2B
  Boling pt:
  Melting pt:
  Solubility:DMSO: 10 mM
  Appearance:Yellow Powder
  Remark:For obtaining a higher solubility , please warm the tube at 37 ˚C and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ˚C for several month.

1. Chen P, et al. J Med Chem. 2015 Apr 6.

• Flow Cytometry (FCM) General Protocol
• Immunofluorescence(IC)
• Immunohistochemistry(Polymer)
• Western Blotting