• Product NameCPI-203
• Brief DescriptionInhibitors
• Purification99.13%
• Biological ActivityCPI-203 is a potent BET bromodomain inhibitor with IC50 of 37 nM for BRD4.
• Target NameEpigenetic Reader Domain inhibitor
• CAS No. 202591-23-9
• Calculated MW 399.9
• Formulation C19H18ClN5OS
• Storage 3 years -20˚C powder;2 years -80˚C in solvent;

• Research Area:Cancer
  SMILES:CC1=C(C)C2=C(S1)N1C(C)=NN=C1C(CC(N)=O)N=C2C1=CC=C(Cl)C=C1
  Pathways:Chromatin/Epigenetic
  Receptor:BRD4
  Boling pt:
  Melting pt:
  Solubility:DMSO: 200 mM
  Appearance:White Powder
  Remark:For obtaining a higher solubility , please warm the tube at 37 ˚C and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ˚C for several month.

1. Devaiah BN, et al. Proc Natl Acad Sci U S A. 2012, 109(18), 6927-6932.

• Flow Cytometry (FCM) General Protocol
• Immunofluorescence(IC)
• Immunohistochemistry(Polymer)
• Western Blotting