• Product NameOrg 27569
• Brief DescriptionInhibitors
• Purification99.50%
• Biological ActivityOrg 27569 is an allosteric modulator of cannabinoid CB1 receptor, induces a CB1 receptor state that is characterized by enhanced agonist affinity and decreased inverse agonist affinity.
• Target NameCannabinoid Receptor modulator
• CAS No. 868273-06-7
• Calculated MW 409.95
• Formulation C24H28ClN3O
• Storage 3 years -20˚C powder;2 years -80˚C in solvent;

• Research Area:Endocrine system
  SMILES:CCC1=C(NC2=C1C=C(Cl)C=C2)C(=O)NCCC1=CC=C(C=C1)N1CCCCC1
  Pathways:GPCR/G Protein
  Receptor:CB1
  Boling pt:
  Melting pt:
  Solubility:DMSO: 82 mg/mL (200.02 mM)
  Appearance:Pink-White Powder
  Remark:For obtaining a higher solubility , please warm the tube at 37 ˚C and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ˚C for several month.

1. Price MR, et al. Mol Pharmacol, 2005, 68(5), 1484-1495.

• Flow Cytometry (FCM) General Protocol
• Immunofluorescence(IC)
• Immunohistochemistry(Polymer)
• Western Blotting