• Product NameDprE1-IN-1
• Brief DescriptionInhibitors
• Purification99.00%
• Biological ActivityDprE1-IN-1 is a potent DprE1 inhibitor, with IC50 of 10 nM, also inhibits PDE6, with IC50 of 6 uM.
• Target NameDprE1 inhibitor
• CAS No. 1494675-86-3
• Calculated MW 355.39
• Formulation C18H21N5O3
• Storage 3 years -20˚C powder;2 years -80˚C in solvent;

• Research Area:Others
  SMILES:CC(=O)C12OC1(C)CC1C3CC=C4CC(O)CCC4(C)C3CCC21C
  Pathways:Others
  Receptor:DprE1
  Boling pt:
  Melting pt:
  Solubility:DMSO: 11 mg/mL
  Appearance:White powder
  Remark:For obtaining a higher solubility , please warm the tube at 37 ˚C and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ˚C for several month.

1. Shirude PS, et al. J Med Chem. 2014 Jul 10;57(13):5728-37.

• Flow Cytometry (FCM) General Protocol
• Immunofluorescence(IC)
• Immunohistochemistry(Polymer)
• Western Blotting