• Product NameGSK-2881078
• Brief DescriptionInhibitors
• Purification98.16%
• Biological ActivityGSK-2881078 is a selective androgen receptor modulator potentially for the treatment of cachexia. GSK2881078 is a selective androgen receptor modulator (SARM) that is being evaluated for effects on muscle growth and strength in subjects with muscle wasting to improve their physical function.
• Target NameAndrogen Receptor inhibitor
• CAS No. 1539314-06-1
• Calculated MW 332.34
• Formulation C14H15F3N2O2S
• Storage 3 years -20˚C powder;2 years -80˚C in solvent;

• Research Area:Nervous system
  SMILES:CC1=C(C(F)(F)F)C2=C(N([C@H](C)CS(=O)(C)=O)CC2)C=C1
  Pathways:Endocrinology/Hormones
  Receptor:Androgen Receptor
  Boling pt:
  Melting pt:
  Solubility:DMSO: 33 mg/mL
  Appearance:White powder
  Remark:For obtaining a higher solubility , please warm the tube at 37 ˚C and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ˚C for several month.

1. GSK-2881078

• Flow Cytometry (FCM) General Protocol
• Immunofluorescence(IC)
• Immunohistochemistry(Polymer)
• Western Blotting