- Product NameRhapontigenin
- Brief DescriptionInhibitors
- Purification99.88%
- Biological ActivityRhapontigenin is a natural analog of resveratrol with antioxidant and anti-cancer activity. It is a mechanism-based, selective inactivator of cytochrome P450 1A1 (IC50?= 400 nM), an aryl hydrocarbon hydroxylase which activates polycyclic aromatic hydrocarbons that act as procarcinogens.1?At higher concentrations, rhapontigenin inhibits the proliferation of HepG2 and HL-60R cancer cell lines (IC50?= 48 μM).
- Target NameP450 inhibitor
- CAS No. 500-65-2
- Calculated MW 258.3
- Formulation C15H14O4
- Storage 3 years -20˚C powder;2 years -80˚C in solvent;