• Product NameGW 501516
• Brief DescriptionInhibitors
• Purification99.00%
• Biological ActivityGW501516 is a potent and highly selective PPARβ/δ agonist, with EC50 of 1 nM, with 1000-fold selectivity over hPPARα and hPPARγ. Phase 4.
• Target NamePPAR agonist
• CAS No. 317318-70-0
• Calculated MW 453.5
• Formulation C21H18F3NO3S2
• Storage 3 years -20˚C powder;2 years -80˚C in solvent;

• Research Area:Cardiovascular system
  SMILES:CC1=C(CSC2=CC(C)=C(OCC(O)=O)C=C2)SC(=N1)C1=CC=C(C=C1)C(F)(F)F
  Pathways:Metabolism
  Receptor:PPARδ
  Boling pt:
  Melting pt:
  Solubility:DMSO>10mMN/AN/A
  Appearance:
  Remark:For obtaining a higher solubility , please warm the tube at 37 ˚C and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ˚C for several month.

1. Sznaidman ML, et al. Bioorg Med Chem Lett, 2003, 13(9), 1517-1521.

• Flow Cytometry (FCM) General Protocol
• Immunofluorescence(IC)
• Immunohistochemistry(Polymer)
• Western Blotting