• Product NameCiproxifan
• Brief DescriptionInhibitors
• Purification98.00%
• Biological ActivityCiproxifan is a highly potent and selective histamin H3-receptor antagonist with IC50 of 9.2 nM, with low apparent affinity at other receptor subtypes.
• Target NameHistamine Receptor antagonist
• CAS No. 184025-18-1
• Calculated MW 386.4
• Formulation C16H18N2O2.C4H4O4
• Storage 3 years -20˚C powder;2 years -80˚C in solvent;

• Research Area:Nervous system
  SMILES:C1CC1C(=O)C2=CC=C(C=C2)OCCCC3=CN=CN3
  Pathways:GPCR/G Protein; Immunology/Inflammation; Neuroscience
  Receptor:H3 receptor
  Boling pt:
  Melting pt:
  Solubility:DMSO:54 mg/mL (139.75 mM)Ethanol:54 mg/mL (139.75 mM)Water:1 mg/mL (2.58 mM)
  Appearance:
  Remark:For obtaining a higher solubility , please warm the tube at 37 ˚C and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ˚C for several month.

1. Ligneau X, et al. J Pharmacol Exp Ther, 1998, 287(2), 658-666.

• Flow Cytometry (FCM) General Protocol
• Immunofluorescence(IC)
• Immunohistochemistry(Polymer)
• Western Blotting