• Product NameTrelagliptin
• Brief DescriptionInhibitors
• Purification98.00%
• Biological ActivityTrelagliptin is a highly selective, long-acting DPP-4 inhibitor. Phase 3.
• Target NameDPP-4 inhibitor
• CAS No. 865759-25-7
• Calculated MW 357.38
• Formulation C18H20FN5O2
• Storage 3 years -20˚C powder;2 years -80˚C in solvent;

• Research Area:Cancer
  SMILES:CN1C(=O)C=C(N(C1=O)CC2=C(C=CC(=C2)F)C#N)N3CCC[C@H](C3)N
  Pathways:Proteases/Proteasome
  Receptor:DPP-4
  Boling pt:
  Melting pt:
  Solubility:Ethanol: 3 mg/mL warmed (8.39 mM); DMSO: 71 mg/mL (198.66 mM)
  Appearance:WhitePowder
  Remark:For obtaining a higher solubility , please warm the tube at 37 ˚C and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ˚C for several month.

1. Inagaki N, et al. Lancet Diabetes Endocrinol. 2014, 2(2), 125-132.

• Flow Cytometry (FCM) General Protocol
• Immunofluorescence(IC)
• Immunohistochemistry(Polymer)
• Western Blotting