• Product NameMozavaptan
• Brief DescriptionInhibitors
• Purification98.00%
• Biological ActivityMozavaptan is a novel competitive vasopressin receptor antagonist for both V1 and V2 receptors with IC50 of 1.2 μM and 14 nM, respectively.
• Target NameVasopressin Receptor antagonist
• CAS No. 137975-06-5
• Calculated MW 427.54
• Formulation C27H29N3O2
• Storage 3 years -20˚C powder;2 years -80˚C in solvent;

• Research Area:Cardiovascular system
  SMILES:CN(C)C1CCCN(C(=O)C2=CC=C(NC(=O)C3=CC=CC=C3C)C=C2)C2=CC=CC=C12
  Pathways:GPCR/G Protein
  Receptor:Vasopressin receptor 1; Vasopressin receptor 2
  Boling pt:
  Melting pt:
  Solubility:DMSO:1 mg/mL (2.33 mM)Ethanol:1 mg/mL (2.33 mM)Water<1 mg/mL (<1 mM)
  Appearance:
  Remark:For obtaining a higher solubility , please warm the tube at 37 ˚C and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ˚C for several month.

1. Burrell LM, et al. Blood Press, 1994, 3(1-2), 137-141.

• Flow Cytometry (FCM) General Protocol
• Immunofluorescence(IC)
• Immunohistochemistry(Polymer)
• Western Blotting