• Product NameFlupirtine maleate
• Brief DescriptionInhibitors
• Purification99.00%
• Biological ActivityFlupirtine maleate is the salt form of Flupirtine, which is a centrally acting non-opioid analgesia, is a selective neuronal potassium channel opener that also has NMDA receptor antagonist properties.
• Target NameNMDAR antagonist; Potassium Channel antagonist
• CAS No. 75507-68-5
• Calculated MW 420.39
• Formulation C15H17FN4O2C4H4O4
• Storage 3 years -20˚C powder;2 years -80˚C in solvent;

• Research Area:Cancer
  SMILES:CCOC(=O)NC1=C(N=C(C=C1)NCC2=CC=C(C=C2)F)N.C(=C\C(=O)O)\C(=O)O
  Pathways:Membrane transporter/Ion channel; Neuroscience
  Receptor:NMDA receptor; Potassium Channel
  Boling pt:
  Melting pt:
  Solubility:Ethanol: 2 mg/mL warmed (4.75 mM); DMSO: 84 mg/mL (199.81 mM)
  Appearance:WhitePowder
  Remark:For obtaining a higher solubility , please warm the tube at 37 ˚C and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ˚C for several month.

1. Perovic S, et al. Eur J Pharmacol, 1994, 288(1), 27-33.

• Flow Cytometry (FCM) General Protocol
• Immunofluorescence(IC)
• Immunohistochemistry(Polymer)
• Western Blotting