• Product NameSGC-CBP30
• Brief DescriptionInhibitors
• Purification99.39%
• Biological ActivitySGC-CBP30 is a potent CREBBP/EP300 inhibitor with IC50 of 21 nM and 38 nM, respectively.
• Target NameEpigenetic Reader Domain inhibitor
• CAS No. 1613695-14-9
• Calculated MW 509.04
• Formulation C28H33CIN4O3
• Storage 3 years -20˚C powder;2 years -80˚C in solvent;

• Research Area:Cancer
  SMILES:CC1=C(C(=NO1)C)C2=CC3=C(C=C2)N(C(=N3)CCC4=CC(=C(C=C4)OC)Cl)C[C@H](C)N5CCOCC5
  Pathways:Chromatin/Epigenetic
  Receptor:CREBBP; EP300
  Boling pt:
  Melting pt:
  Solubility:Ethanol: 100 mg/mL (196.44 mM); DMSO: 100 mg/mL (196.44 mM)
  Appearance:
  Remark:For obtaining a higher solubility , please warm the tube at 37 ˚C and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ˚C for several month.

1. Structural Genomics Consortium

• Flow Cytometry (FCM) General Protocol
• Immunofluorescence(IC)
• Immunohistochemistry(Polymer)
• Western Blotting