• Product NameSB366791
• Brief DescriptionInhibitors
• Purification98.00%
• Biological ActivitySB-366791 is a novel, potent, and selective, cinnamide TRPV1 antagonist.
• Target NameTRP/TRPV Channel inhibitor
• CAS No. 472981-92-3
• Calculated MW 287.74
• Formulation C16H14ClNO2
• Storage 3 years -20˚C powder;2 years -80˚C in solvent;

• Research Area:Others
  SMILES:COC1=CC=CC(=C1)NC(=O)/C=C/C2=CC=C(C=C2)Cl
  Pathways:Membrane transporter/Ion channel
  Receptor:TRPV1
  Boling pt:
  Melting pt:
  Solubility:Ethanol: <1 mg/mLDMSO: 57 mg/mL (198.09 mM) Water: <1 mg/mL
  Appearance:
  Remark:For obtaining a higher solubility , please warm the tube at 37 ˚C and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ˚C for several month.

1. Gunthorpe MJ,et al. Identification and characterisation of SB-366791, a potent and selective vanilloid receptor (VR1/TRPV1) antagonist. Neuropharmacology. 2004 Jan;46(1):133-49.

• Flow Cytometry (FCM) General Protocol
• Immunofluorescence(IC)
• Immunohistochemistry(Polymer)
• Western Blotting